SCHEMBL9705898

SCHEMBL9705898

Cc1cc(CCCCCOc2c(Cl)cc(C(=O)O)cc2C(F)(F)F)on1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
PLAU P00749 1/20 0.39
MRGPRX4 Q96LA9 4/20 0.33
HDAC6 Q9UBN7 1/20 0.33
PPARG P37231 1/20 0.33
RORC P51449 1/20 0.33
RARB P10826 2/20 0.33
PLA2G2A P14555 2/20 0.33
KDM4C Q9H3R0 1/20 0.33
RARA P10276 1/20 0.33
RARG P13631 1/20 0.33
PPARA Q07869 1/20 0.33
TPMT P51580 1/20 0.33
POLB P06746 1/20 0.32
ALOX15 P16050 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9200429 0.90 PLAU (0.49) NR1I2CYP3A4CYP2D6PLAUMRGPRX4
SCHEMBL9706268 0.86 NR1I2 (0.45) NR1I2CYP3A4CYP2D6PLAUMRGPRX4
SCHEMBL10413141 0.85 PLAU (0.51) NR1I2CYP3A4CYP2D6PLAUHDAC6
SCHEMBL9706270 0.85 KDM4E (0.42) NR1I2CYP3A4CYP2D6PLAUHDAC6
SCHEMBL9705949 0.81 TPMT (0.39) NR1I2CYP3A4CYP2D6PLAUTPMT
SCHEMBL9705668 0.81 NR1I2 (0.45) NR1I2CYP3A4CYP2D6
SCHEMBL9862923 0.81 NR1I2 (0.45) NR1I2CYP3A4CYP2D6PLAURARB
SCHEMBL9436198 0.80 LMNA (0.42) NR1I2CYP3A4CYP2D6PLAUHDAC6
SCHEMBL9705669 0.79 CYP2D6 (0.41) NR1I2CYP3A4CYP2D6PLAUMRGPRX4
SCHEMBL9863245 0.78 POLB (0.45) NR1I2CYP3A4CYP2D6TPMTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0207454-B1 ISOXAZOLE AND FURAN DERIVATIVES, THEIR PREPARATION AND USE AS ANTIVIRAL AGENTS STERLING WINTHROP INC. (US) 1992-09-09 EP disclosed
US-5002960-A Viricides for combating picornaviruses STERLING DRUG, INC. (US) 1991-03-26 US disclosed
US-4939267-A Viricides STERLING DRUG INC. (US) 1990-07-03 US disclosed
US-4843087-A OXAZOLINYL COMPOUNDS; RHINOVIRUSES AND PICORNAVIRUSES STERLING DRUG INC. (US) 1989-06-27 US disclosed
EP-0207454-A2 Isoxazole and furan derivatives, their preparation and use as antiviral agents STERLING WINTHROP INC. (US) 1987-01-07 EP disclosed