SCHEMBL9705877

SCHEMBL9705877

O=C1Nc2cccnc2N(c2ccccc2)c2ncccc21

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
RAB9A P51151 1/20 0.50
ALDH1A1 P00352 2/20 0.47
ALOX15 P16050 1/20 0.47
MAPK10 P53779 1/20 0.47
HSD17B10 Q99714 1/20 0.47
LMNA P02545 2/20 0.43
CHRM2 P08172 2/20 0.43
USP2 O75604 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CYP2D6 P10635 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
GMNN O75496 1/20 0.42
APEX1 P27695 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300867 0.76 RAB9A (0.53) CYP1A2SMN1; SMN2RAB9AALDH1A1ALOX15
SCHEMBL8300334 0.73 RAB9A (0.50) CYP1A2SMN1; SMN2RAB9AALDH1A1ALOX15
SCHEMBL8304745 0.73 CYP1A2 (0.49) CYP1A2SMN1; SMN2RAB9AALDH1A1ALOX15
SCHEMBL8790773 0.73 RAB9A (0.53) CYP1A2SMN1; SMN2RAB9AALDH1A1LMNA
SCHEMBL9174480 0.73 RAB9A (0.60) CYP1A2SMN1; SMN2RAB9AALDH1A1LMNA
SCHEMBL9705864 0.72 RAB9A (0.58) CYP1A2RAB9AALDH1A1LMNACHRM2
SCHEMBL8889164 0.72 BRD4 (0.44) SMN1; SMN2ALDH1A1HSD17B10
SCHEMBL9704493 0.72 ALDH1A1 (0.70) CYP1A2SMN1; SMN2RAB9AALDH1A1ALOX15
SCHEMBL8301869 0.71 CHRM2 (0.48) CYP1A2SMN1; SMN2RAB9AALDH1A1LMNA
SCHEMBL11202566 0.71 RAB9A (0.66) CYP1A2RAB9AALDH1A1LMNACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0482481-A1 Method for the preparation of 5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepines BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1992-04-29 EP disclosed