SCHEMBL9707286

SCHEMBL9707286

CCCCc1nc2c(c(=O)[nH]c(=O)n2CCC)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 9/20 0.50
AGTR2 P50052 9/20 0.50
TPH1 P17752 3/20 0.49
TPH2 Q8IWU9 3/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708233 0.98 TPH1 (0.49) AGTR1AGTR2TPH1TPH2MEN1
SCHEMBL9708270 0.95 MEN1 (0.49) AGTR1AGTR2TPH1TPH2MEN1
SCHEMBL9707811 0.95 TPH1 (0.51) AGTR1AGTR2TPH1TPH2MEN1
SCHEMBL9708426 0.94 MEN1 (0.53) AGTR1AGTR2TPH1TPH2MEN1
SCHEMBL9707594 0.93 AGTR1 (0.47) AGTR1AGTR2MEN1KMT2AALDH1A1
SCHEMBL9708208 0.93 ALDH1A1 (0.49) AGTR1AGTR2TPH1TPH2MEN1
SCHEMBL9707992 0.93 USP2 (0.51) AGTR1AGTR2MEN1KMT2AALDH1A1
SCHEMBL9708861 0.93 TPH1 (0.51) AGTR1AGTR2TPH1TPH2MEN1
SCHEMBL9707289 0.92 MEN1 (0.52) AGTR1AGTR2TPH1TPH2MEN1
SCHEMBL9707854 0.91 AGTR1 (0.48) AGTR1AGTR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO claimed
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed