SCHEMBL9707745

SCHEMBL9707745

CCn1c(=O)c2c(nc(C(C)C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(CCOC)c1=O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.39
ADORA2B P29275 2/20 0.39
ADORA3 P0DMS8 4/20 0.39
USP1 O94782 2/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PKM P14618 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ADORA1 P30542 3/20 0.36
DCTPP1 Q9H773 1/20 0.36
TSHR P16473 1/20 0.36
PDE5A O76074 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707692 0.98 ADORA3 (0.40) ADORA2AADORA2BADORA3USP1KDM4E
SCHEMBL9707871 0.96 ADORA3 (0.42) ADORA2AADORA2BADORA3USP1KDM4E
SCHEMBL9707508 0.95 ADORA3 (0.42) ADORA2AADORA2BADORA3USP1ADORA1
SCHEMBL9707777 0.95 ADORA3 (0.42) ADORA2AADORA2BADORA3USP1ADORA1
SCHEMBL9708054 0.93 USP1 (0.42) ADORA3USP1ALDH1A1MEN1KMT2A
SCHEMBL9708350 0.92 ADORA3 (0.43) ADORA2AADORA2BADORA3ADORA1
SCHEMBL9707419 0.92 ADORA3 (0.42) ADORA2AADORA2BADORA3USP1KDM4E
SCHEMBL9708021 0.92 ADORA3 (0.42) ADORA2AADORA2BADORA3USP1KDM4E
SCHEMBL9707864 0.91 DCTPP1 (0.46) USP1MEN1KMT2ADCTPP1
SCHEMBL9708822 0.90 KMT2A (0.40) ADORA3USP1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed