SCHEMBL9707777

SCHEMBL9707777

CCCn1c(=O)n(CCOC)c(=O)c2c1nc(C(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 15/20 0.42
ADORA1 P30542 4/20 0.42
ADORA2B P29275 3/20 0.39
ADORA2A P29274 2/20 0.39
USP1 O94782 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707508 1.00 ADORA3 (0.42) ADORA3ADORA1ADORA2BADORA2AUSP1
SCHEMBL9707871 0.97 ADORA3 (0.42) ADORA3ADORA1ADORA2BADORA2AUSP1
SCHEMBL9707692 0.95 ADORA3 (0.40) ADORA3ADORA1ADORA2BADORA2AUSP1
SCHEMBL9707745 0.95 ADORA2A (0.39) ADORA3ADORA1ADORA2BADORA2AUSP1
SCHEMBL9707739 0.94 ADORA3 (0.47) ADORA3ADORA1ADORA2BADORA2A
SCHEMBL9708021 0.92 ADORA3 (0.42) ADORA3ADORA1ADORA2BADORA2AUSP1
SCHEMBL9707419 0.92 ADORA3 (0.42) ADORA3ADORA1ADORA2BADORA2AUSP1
SCHEMBL9707864 0.92 DCTPP1 (0.46) USP1
SCHEMBL9708054 0.92 USP1 (0.42) ADORA3USP1
SCHEMBL9708350 0.91 ADORA3 (0.43) ADORA3ADORA1ADORA2BADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed