SCHEMBL9707519

SCHEMBL9707519

CC(C)Cn1c(=O)c2c(nc(C(C)C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(-c2ccccc2)c1=O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.39
ADORA1 P30542 4/20 0.39
ADORA2A P29274 2/20 0.36
ADORA2B P29275 2/20 0.36
AGTR1 P30556 1/20 0.36
AGTR2 P50052 1/20 0.36
USP1 O94782 1/20 0.35
RAB9A P51151 1/20 0.35
PDE4A P27815 1/20 0.35
KMT2A Q03164 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707604 0.94 ADORA1 (0.37) ADORA3ADORA1ADORA2AADORA2BAGTR1
SCHEMBL9707906 0.93 AGTR1 (0.38) ADORA3ADORA1ADORA2AAGTR1AGTR2
SCHEMBL9708160 0.92 AGTR1 (0.37) AGTR1AGTR2USP1
SCHEMBL9708757 0.91 ADORA3 (0.41) ADORA3ADORA1ADORA2AADORA2BAGTR1
SCHEMBL9708737 0.91 ADORA3 (0.40) ADORA3ADORA1ADORA2AADORA2BAGTR1
SCHEMBL9708819 0.91 ADORA3 (0.44) ADORA3ADORA1ADORA2AADORA2BAGTR1
SCHEMBL9707898 0.91 MAPT (0.38) ADORA3ADORA1AGTR1AGTR2USP1
SCHEMBL9707660 0.90 USP1 (0.39) AGTR1AGTR2USP1
SCHEMBL9707563 0.90 AGTR1 (0.41) ADORA3ADORA1AGTR1AGTR2
SCHEMBL9707347 0.90 RAB9A (0.44) ADORA3ADORA1ADORA2AADORA2BUSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed