SCHEMBL9707553

SCHEMBL9707553

CCc1nc2c(c(=O)n(C)c(=O)n2CC(C)C)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 1/20 0.43
PDE1B Q01064 1/20 0.43
PDE1C Q14123 1/20 0.43
AGTR1 P30556 1/20 0.42
AGTR2 P50052 1/20 0.42
NPSR1 Q6W5P4 3/20 0.41
TSHR P16473 3/20 0.41
LMNA P02545 2/20 0.41
CASP1 P29466 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HSD17B10 Q99714 2/20 0.41
ALOX15 P16050 1/20 0.41
PDE5A O76074 6/20 0.41
HTT P42858 2/20 0.41
CASP7 P55210 1/20 0.41
ALDH1A1 P00352 2/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708190 0.94 AGTR1 (0.43) PDE1APDE1BPDE1CAGTR1AGTR2
SCHEMBL9708497 0.93 RAB9A (0.43) AGTR1AGTR2NPSR1TSHRLMNA
SCHEMBL9708698 0.93 ADORA3 (0.43) AGTR1AGTR2
SCHEMBL9707555 0.92 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL9708105 0.92 ADORA3 (0.42) AGTR1AGTR2
SCHEMBL9707700 0.92 AGTR1 (0.42) AGTR1AGTR2
SCHEMBL9707579 0.92 AGTR1 (0.44) AGTR1AGTR2NPSR1TSHRHSD17B10
SCHEMBL9707554 0.91 AGTR1 (0.45) AGTR1AGTR2PDE5A
SCHEMBL9709079 0.91 PDE1A (0.43) PDE1APDE1BPDE1CNPSR1TSHR
SCHEMBL9708492 0.91 AGTR1 (0.41) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed