SCHEMBL9707579

SCHEMBL9707579

CCc1nc2c(c(=O)n(C)c(=O)n2CC)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 5/20 0.44
AGTR2 P50052 5/20 0.44
ALOX15 P16050 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
HTT P42858 1/20 0.42
TSHR P16473 1/20 0.42
HPGD P15428 1/20 0.42
GPR18 Q14330 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707817 0.94 AGTR1 (0.44) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9708564 0.93 AGTR1 (0.46) AGTR1AGTR2ALOX15HSD17B10
SCHEMBL9708840 0.93 AGTR1 (0.44) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9707699 0.93 ALOX15 (0.52) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9707475 0.92 ALOX15 (0.41) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9707540 0.92 AGTR1 (0.50) AGTR1AGTR2
SCHEMBL9708268 0.92 TSHR (0.46) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9707553 0.92 PDE1A (0.43) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9708324 0.91 ADORA3 (0.43) AGTR1AGTR2
SCHEMBL9707744 0.91 AGTR1 (0.48) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed