SCHEMBL9707609

SCHEMBL9707609

COCCn1c(=O)n(-c2ccccc2)c(=O)c2c1nc(C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DCTPP1 Q9H773 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
BRD4 O60885 1/20 0.36
GAA P10253 1/20 0.36
RECQL P46063 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
AGTR1 P30556 2/20 0.35
AGTR2 P50052 2/20 0.35
PPARG P37231 1/20 0.35
NSD2 O96028 1/20 0.35
IDO1 P14902 1/20 0.35
CRHBP P24387 1/20 0.35
TDO2 P48775 1/20 0.35
CASP7 P55210 1/20 0.35
CASP6 P55212 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708557 0.94 DCTPP1 (0.43) DCTPP1KDM4EALDH1A1PKMADORA3
SCHEMBL9708509 0.91 ADORA3 (0.40) ADORA3AGTR1AGTR2
SCHEMBL9708369 0.91 AGTR1 (0.39) MEN1KMT2AAGTR1AGTR2
SCHEMBL9708117 0.90 DCTPP1 (0.43) DCTPP1KDM4EALDH1A1PKMADORA3
SCHEMBL9708900 0.90 USP1 (0.39) DCTPP1KDM4EALDH1A1PKMADORA3
SCHEMBL9707578 0.90 DCTPP1 (0.41) DCTPP1KDM4EALDH1A1PKMADORA3
SCHEMBL9707722 0.90 AGTR1 (0.39) ALDH1A1ADORA3AGTR1AGTR2
SCHEMBL9708091 0.89 AGTR1 (0.41) AGTR1AGTR2
SCHEMBL9708292 0.89 ADORA3 (0.42) DCTPP1ADORA3
SCHEMBL9707598 0.89 DCTPP1 (0.42) DCTPP1KDM4EALDH1A1PKMADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed