SCHEMBL9707828

SCHEMBL9707828

Cc1nc2c(c(=O)[nH]c(=O)n2-c2ccccc2)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.42
ALDH1A1 P00352 5/20 0.42
HTT P42858 3/20 0.42
MAPT P10636 3/20 0.42
HPGD P15428 2/20 0.42
GAA P10253 1/20 0.42
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
NPSR1 Q6W5P4 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 3/20 0.39
PKM P14618 2/20 0.39
MCL1 Q07820 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
AGTR1 P30556 1/20 0.39
AGTR2 P50052 1/20 0.39
BRAF P15056 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CXCL8 P10145 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708587 0.90 AGTR1 (0.45) KDM4EALDH1A1HTTMAPTHPGD
SCHEMBL9708009 0.89 CXCL8 (0.39) KDM4EALDH1A1HTTMAPTHPGD
SCHEMBL9708366 0.88 BRAF (0.48) KDM4EALDH1A1HTTMAPTHPGD
SCHEMBL9707926 0.88 AGTR2 (0.46) MEN1KMT2AAGTR1AGTR2
SCHEMBL9707767 0.88 MEN1 (0.50) KDM4EALDH1A1HTTMAPTHPGD
SCHEMBL9708221 0.88 MEN1 (0.41) KDM4EALDH1A1HTTMAPTHPGD
SCHEMBL9707732 0.87 ALDH1A1 (0.47) KDM4EALDH1A1HTTMAPTHPGD
SCHEMBL9707742 0.87 AGTR2 (0.49) AGTR1AGTR2
SCHEMBL9707935 0.87 AGTR1 (0.39) ALDH1A1AGTR1AGTR2
SCHEMBL9708479 0.86 AGTR2 (0.46) MEN1KMT2AAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed