SCHEMBL9707973

SCHEMBL9707973

CC(C)Cn1c(=O)c2c(nc(CC(C)(C)C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(CCc2ccccc2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.42
ADORA3 P0DMS8 4/20 0.42
AGTR1 P30556 5/20 0.38
AGTR2 P50052 2/20 0.38
LMNA P02545 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
ADORA2A P29274 2/20 0.37
ADORA2B P29275 2/20 0.37
MAPK1 P28482 1/20 0.37
TSHR P16473 1/20 0.36
CASP1 P29466 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RAB9A P51151 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707877 0.94 AGTR1 (0.42) ADORA1ADORA3AGTR1AGTR2NPSR1
SCHEMBL9708158 0.94 ADORA3 (0.41) ADORA1ADORA3AGTR1AGTR2ADORA2A
SCHEMBL9708090 0.93 ADORA3 (0.39) ADORA1ADORA3AGTR1AGTR2ADORA2A
SCHEMBL9707495 0.92 ADORA1 (0.45) ADORA1ADORA3AGTR1AGTR2ADORA2A
SCHEMBL9708576 0.92 ADORA1 (0.40) ADORA1ADORA3AGTR1AGTR2ADORA2A
SCHEMBL9708732 0.92 ADORA3 (0.43) ADORA1ADORA3AGTR1AGTR2
SCHEMBL9707297 0.91 ADORA3 (0.43) ADORA1ADORA3AGTR1AGTR2ADORA2A
SCHEMBL9708598 0.91 ADORA1 (0.44) ADORA1ADORA3AGTR1AGTR2ADORA2A
SCHEMBL9707529 0.91 ADORA3 (0.43) ADORA1ADORA3AGTR1AGTR2ADORA2A
SCHEMBL9707531 0.91 ADORA1 (0.43) ADORA1ADORA3AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed