SCHEMBL9707495

SCHEMBL9707495

CCn1c(=O)c2c(nc(CC(C)(C)C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(CCc2ccccc2)c1=O

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.45
AGTR1 P30556 5/20 0.41
ADORA2A P29274 3/20 0.41
AGTR2 P50052 3/20 0.41
ADORA2B P29275 2/20 0.41
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
PDE5A O76074 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708598 0.98 ADORA1 (0.44) ADORA1AGTR1ADORA2AAGTR2ADORA2B
SCHEMBL9707877 0.96 AGTR1 (0.42) ADORA1AGTR1AGTR2HSD17B10ADORA3
SCHEMBL9707297 0.95 ADORA3 (0.43) ADORA1AGTR1ADORA2AAGTR2ADORA2B
SCHEMBL9707529 0.95 ADORA3 (0.43) ADORA1AGTR1ADORA2AAGTR2ADORA2B
SCHEMBL9708161 0.94 ADORA1 (0.43) ADORA1AGTR1ADORA2AAGTR2ADORA2B
SCHEMBL9707632 0.93 ALOX15 (0.43) AGTR1AGTR2TSHRHSD17B10
SCHEMBL9708004 0.93 ADORA3 (0.40) ADORA1AGTR1ADORA2AAGTR2ADORA2B
SCHEMBL9707629 0.92 ADORA1 (0.48) ADORA1AGTR1ADORA2AAGTR2ADORA2B
SCHEMBL9707973 0.92 ADORA1 (0.42) ADORA1AGTR1ADORA2AAGTR2ADORA2B
SCHEMBL9708387 0.92 POLB (0.44) AGTR1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed