SCHEMBL9707877

SCHEMBL9707877

CC(C)(C)Cc1nc2c(c(=O)n(CCc3ccccc3)c(=O)n2CCc2ccccc2)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 7/20 0.42
AGTR2 P50052 3/20 0.41
POLB P06746 1/20 0.40
HIF1A Q16665 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ADORA1 P30542 1/20 0.39
ALOX15 P16050 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HSD17B10 Q99714 1/20 0.39
TP53 P04637 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708598 0.97 ADORA1 (0.44) AGTR1AGTR2ADORA1HSD17B10ADORA3
SCHEMBL9707297 0.97 ADORA3 (0.43) AGTR1AGTR2ADORA1ADORA3
SCHEMBL9707529 0.97 ADORA3 (0.43) AGTR1AGTR2ADORA1ADORA3
SCHEMBL9707495 0.96 ADORA1 (0.45) AGTR1AGTR2ADORA1HSD17B10ADORA3
SCHEMBL9708387 0.95 POLB (0.44) AGTR1POLBHIF1AALOX15ALDH1A1
SCHEMBL9707632 0.95 ALOX15 (0.43) AGTR1AGTR2ALOX15ALDH1A1HSD17B10
SCHEMBL9708824 0.95 ADORA3 (0.41) AGTR1AGTR2MEN1KMT2AALDH1A1
SCHEMBL9708259 0.95 ADORA3 (0.41) AGTR1AGTR2MEN1KMT2AALDH1A1
SCHEMBL9707973 0.94 ADORA1 (0.42) AGTR1AGTR2MEN1KMT2AADORA1
SCHEMBL9708814 0.93 AGTR1 (0.39) AGTR1AGTR2POLBHIF1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed