SCHEMBL9708124

SCHEMBL9708124

CCCc1nc2c(c(=O)[nH]c(=O)n2CC)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
TPH1 P17752 17/20 0.49
TPH2 Q8IWU9 17/20 0.49
AGTR1 P30556 1/20 0.48
AGTR2 P50052 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708426 0.95 MEN1 (0.53) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9707289 0.94 MEN1 (0.52) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9707811 0.94 TPH1 (0.51) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9708297 0.93 MEN1 (0.54) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9708930 0.93 MEN1 (0.50) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9708184 0.92 MEN1 (0.47) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9708629 0.91 AGTR1 (0.48) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9707568 0.90 ALDH1A1 (0.48) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9708379 0.90 MEN1 (0.46) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9707269 0.90 MEN1 (0.51) MEN1KMT2ATPH1TPH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed