SCHEMBL9708253

SCHEMBL9708253

COC(C)n1c(=O)c2c(nc(C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(CC(C)C)c1=O

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.36
ADORA3 P0DMS8 2/20 0.36
AGTR1 P30556 2/20 0.36
AGTR2 P50052 2/20 0.36
ADORA1 P30542 2/20 0.35
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708428 0.94 ADORA3 (0.38) PDE5AADORA3AGTR1AGTR2ADORA1
SCHEMBL9707596 0.93 AGTR1 (0.36) AGTR1AGTR2
SCHEMBL9708661 0.93 AGTR1 (0.38) AGTR1AGTR2
SCHEMBL9707503 0.91 ADORA3 (0.38) ADORA3ADORA1ADORA2B
SCHEMBL9708025 0.91 AGTR1 (0.40) AGTR1AGTR2
SCHEMBL9707571 0.90 ALDH1A1 (0.38) AGTR1AGTR2
SCHEMBL9707684 0.90 ADORA1 (0.37) ADORA3AGTR1AGTR2ADORA1ADORA2A
SCHEMBL9708665 0.90 AGTR1 (0.38) AGTR1AGTR2
SCHEMBL9707395 0.89 PDE5A (0.41) PDE5AADORA3AGTR1AGTR2ADORA2A
SCHEMBL9707855 0.89 AGTR1 (0.39) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed