SCHEMBL9708311

SCHEMBL9708311

CCn1c(=O)n(CC(C)C)c(=O)c2c1nc(C(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.42
ADORA3 P0DMS8 5/20 0.42
ADORA2A P29274 4/20 0.38
ADORA2B P29275 3/20 0.38
AGTR1 P30556 1/20 0.37
PDE5A O76074 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708431 0.97 ADORA1 (0.40) ADORA1ADORA3ADORA2AADORA2BPDE5A
SCHEMBL9708819 0.96 ADORA3 (0.44) ADORA1ADORA3ADORA2AADORA2BAGTR1
SCHEMBL9708654 0.94 ADORA3 (0.42) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL9707841 0.92 ADORA3 (0.44) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL9707347 0.91 RAB9A (0.44) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL9708350 0.91 ADORA3 (0.43) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL9708826 0.90 HPGD (0.41)
SCHEMBL9708048 0.90 PDE5A (0.44) ADORA1ADORA3ADORA2AAGTR1PDE5A
SCHEMBL9707502 0.90 ADORA1 (0.42) ADORA1ADORA3ADORA2AAGTR1PDE5A
SCHEMBL9708391 0.89 PDE1A (0.44) PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed