SCHEMBL9708857

SCHEMBL9708857

CC(C)c1nc2c(c(=O)[nH]c(=O)n2CC2CC2)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 4/20 0.39
HTT P42858 3/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 2/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 7/20 0.39
MEN1 O00255 6/20 0.39
NPSR1 Q6W5P4 4/20 0.39
TSHR P16473 2/20 0.38
AGTR1 P30556 1/20 0.38
AGTR2 P50052 1/20 0.38
CXCL8 P10145 1/20 0.38
NOD2 Q9HC29 1/20 0.38
NOD1 Q9Y239 1/20 0.38
PKM P14618 1/20 0.38
MCL1 Q07820 1/20 0.38
HSD17B10 Q99714 1/20 0.38
USP1 O94782 2/20 0.37
POLB P06746 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708645 0.90 ALDH1A1 (0.42) ALDH1A1KDM4EHTTMAPTHPGD
SCHEMBL9707643 0.89 MEN1 (0.48) ALDH1A1KDM4EHTTMAPTHPGD
SCHEMBL9707557 0.89 ALDH1A1 (0.43) ALDH1A1KDM4EHTTMAPTHPGD
SCHEMBL9707980 0.88 PDE5A (0.49) AGTR1AGTR2PDE5APDE4APDE4B
SCHEMBL9708230 0.88 KMT2A (0.45) ALDH1A1KDM4EHTTMAPTHPGD
SCHEMBL9707464 0.88 MEN1 (0.45) ALDH1A1KDM4EHTTMAPTHPGD
SCHEMBL9707357 0.87 ADORA2A (0.41) AGTR1AGTR2USP1PDE5APDE4A
SCHEMBL9708303 0.87 ALDH1A1 (0.44) ALDH1A1KDM4EHTTMAPTHPGD
SCHEMBL9708130 0.87 CXCL8 (0.49) ALDH1A1KDM4EHTTMAPTHPGD
SCHEMBL9708133 0.87 PDE5A (0.41) ALDH1A1HPGDNPSR1TSHRAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed