SCHEMBL9708130

SCHEMBL9708130

CC(C)c1nc2c(c(=O)[nH]c(=O)n2C)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCL8 P10145 2/20 0.49
NOD2 Q9HC29 2/20 0.49
NOD1 Q9Y239 2/20 0.49
ALDH1A1 P00352 5/20 0.46
TSHR P16473 4/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
HPGD P15428 2/20 0.46
MAPK1 P28482 2/20 0.46
BRAF P15056 1/20 0.46
POLB P06746 3/20 0.45
HTT P42858 2/20 0.45
KDM4E B2RXH2 1/20 0.45
TNF P01375 1/20 0.45
MAPT P10636 1/20 0.45
G6PD P11413 1/20 0.45
RAB9A P51151 1/20 0.45
PAX8 Q06710 1/20 0.45
TLR9 Q9NR96 1/20 0.45
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707464 0.91 MEN1 (0.45) CXCL8NOD2NOD1ALDH1A1TSHR
SCHEMBL9707643 0.90 MEN1 (0.48) CXCL8NOD2NOD1ALDH1A1TSHR
SCHEMBL9708303 0.90 ALDH1A1 (0.44) CXCL8NOD2NOD1ALDH1A1TSHR
SCHEMBL9707557 0.90 ALDH1A1 (0.43) CXCL8NOD2NOD1ALDH1A1TSHR
SCHEMBL9708009 0.89 CXCL8 (0.39) CXCL8NOD2NOD1ALDH1A1TSHR
SCHEMBL9707717 0.88 ALDH1A1 (0.49) ALDH1A1MEN1KMT2AHPGDMAPK1
SCHEMBL9708366 0.88 BRAF (0.48) CXCL8NOD2NOD1ALDH1A1TSHR
SCHEMBL9707712 0.88 KDM4E (0.40) CXCL8NOD2NOD1ALDH1A1TSHR
SCHEMBL9708293 0.88 USP1 (0.39) CXCL8NOD2NOD1ALDH1A1TSHR
SCHEMBL9708857 0.87 ALDH1A1 (0.39) CXCL8NOD2NOD1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed