SCHEMBL9709971

SCHEMBL9709971

Cc1cc(NCc2ccc(-c3ccccc3C(=O)O)cc2)c2nc(C(N)=O)ccc2n1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CD38 P28907 9/20 0.52
BDKRB1 P46663 1/20 0.43
AGTR2 P50052 2/20 0.42
LTB4R2 Q9NPC1 1/20 0.41
VCP P55072 1/20 0.41
AGTR1 P30556 1/20 0.41
OPRL1 P41146 1/20 0.41
CYP3A4 P08684 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9709799 0.93 CD38 (0.47) CD38BDKRB1AGTR2LTB4R2VCP
SCHEMBL9709814 0.84 CD38 (0.55) CD38BDKRB1VCP
SCHEMBL9709809 0.82 AGTR1 (0.45) CD38AGTR2AGTR1
SCHEMBL3058636 0.82 CD38 (0.56) CD38BDKRB1LTB4R2
Hydrochloric Acid SCHEMBL9494706 0.81 CD38 (0.55) CD38BDKRB1LTB4R2
SCHEMBL9709869 0.81 AGTR1 (0.43) CD38BDKRB1AGTR2LTB4R2VCP
SCHEMBL9709700 0.81 VCP (0.52) CD38BDKRB1AGTR2VCPAGTR1
SCHEMBL9709660 0.80 AGTR1 (0.45) AGTR2LTB4R2AGTR1
SCHEMBL9709608 0.78 CD38 (0.50) CD38BDKRB1AGTR2LTB4R2VCP
SCHEMBL9709886 0.78 AGTR1 (0.46) CD38AGTR2VCPAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992022533-A1 4-AMINOQUINOLINES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UPJOHN COMPANY (US) 1992-12-23 WO claimed
WO-1992022533-A1 4-AMINOQUINOLINES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UPJOHN COMPANY (US) 1992-12-23 WO disclosed