SCHEMBL9710360

SCHEMBL9710360

CC(=O)n1c(N)nc2nc[nH]c2c1=O.Nc1nc(SCc2ccccc2)c2[nH]cnc2n1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.68
POLB P06746 1/20 0.68
CYP1A2 P05177 7/20 0.55
CYP3A4 P08684 6/20 0.55
CYP2C19 P33261 6/20 0.55
CYP2D6 P10635 4/20 0.55
CYP2C9 P11712 4/20 0.55
NUDT1 P36639 2/20 0.55
ALDH1A1 P00352 2/20 0.55
HIF1A Q16665 2/20 0.55
TOP2A P11388 1/20 0.55
HPGD P15428 1/20 0.55
HSD17B10 Q99714 1/20 0.55
ENPP1 P22413 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.48
CDC7 O00311 2/20 0.46
DBF4 Q9UBU7 2/20 0.46
MAP3K5 Q99683 1/20 0.42
CDK1 P06493 3/20 0.42
CDK2 P24941 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2115657 0.82 PIN1 (1.00) PIN1POLBCYP1A2CYP3A4CYP2C19
Benzene SCHEMBL8024450 0.81 MGMT (0.43) CYP1A2CYP2C19ALDH1A1HSD17B10ENPP1
SCHEMBL218669 0.79 MGMT (0.45) CYP1A2CYP2C19ALDH1A1HIF1AHSD17B10
Bromide SCHEMBL8165615 0.78 MGMT (0.44) CYP1A2CYP2C19ALDH1A1HIF1AHSD17B10
SCHEMBL3305057 0.76 PIN1 (0.76) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL28368763 0.75 PNP (0.45) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL25398225 0.73 LMNA (0.53) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL8583450 0.72 CDK1 (0.49) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL24846529 0.72 POLB (0.78) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL24846512 0.72 CYP1A2 (1.00) PIN1POLBCYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992020816-A1 DETERMINATION OF PRODRUGS METABOLIZABLE BY THE LIVER AND THERAPEUTIC USE THEREOF YALE UNIVERSITY (US) 1992-11-26 WO disclosed