SCHEMBL9711196

SCHEMBL9711196

O=[N+]([O-])CSc1cccc2ccc(Cl)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PDE7A Q13946 9/20 0.39
TDP1 Q9NUW8 1/20 0.37
PDE7B Q9NP56 3/20 0.36
CYP2A6 P11509 1/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
CCR2 P41597 1/20 0.33
FBP1 P09467 1/20 0.33
HPRT1 P00492 1/20 0.33
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27051255 0.72 CYP2A6 (0.45) ALDH1A1MEN1KMT2ACYP2A6
SCHEMBL12728634 0.71 ALDH1A1 (0.61) ALDH1A1MEN1KMT2APDE7ATDP1
SCHEMBL9740858 0.71 USP7 (0.42) ALDH1A1MEN1KMT2APDE7ATDP1
SCHEMBL9739624 0.71 LMNA (0.46) ALDH1A1MEN1KMT2APDE7ATDP1
SCHEMBL9711256 0.70 KIF18A (0.37) ALDH1A1TDP1CYP2A6MAPTTSHR
SCHEMBL9711238 0.70 CYP2A6 (0.37) ALDH1A1MEN1KMT2ATDP1CYP2A6
SCHEMBL9711273 0.69 KMT2A (0.37) ALDH1A1MEN1KMT2APDE7ATDP1
SCHEMBL9711280 0.69 CYP3A4 (0.44) ALDH1A1MEN1KMT2ATDP1TSHR
SCHEMBL9711236 0.69 TDP1 (0.40) ALDH1A1MEN1KMT2APDE7ATDP1
SCHEMBL15352079 0.68 CYP2A6 (0.48) MEN1KMT2ACYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5153227-A Treatment of diabetes and galactosemia complications IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-10-06 US disclosed
EP-0304190-B1 (ARYLSULPHONYL)NITROMETHANES, PROCESS FOR THEIR PREPARATION AND USE IN PHARMACEUTICAL COMPOSITIONS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-07-08 EP disclosed
EP-0304190-A1 (Arylsulphonyl)nitromethanes, process for their preparation and use in pharmaceutical compositions IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-02-22 EP disclosed