SCHEMBL9713813

SCHEMBL9713813

COC(=O)c1cc(N)ccc1S(=O)(=O)c1ccc(NC(C)=O)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.67
PKM P14618 3/20 0.62
CYP2C19 P33261 1/20 0.62
GAA P10253 2/20 0.51
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 3/20 0.50
HPGD P15428 2/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50
HSD17B10 Q99714 1/20 0.50
CA1 P00915 3/20 0.48
CA2 P00918 3/20 0.48
CA12 O43570 2/20 0.48
CA9 Q16790 2/20 0.48
SMN1; SMN2 Q16637 4/20 0.47
LMNA P02545 2/20 0.46
NPC1 O15118 1/20 0.46
F2 P00734 1/20 0.46
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713853 0.88 PKM (0.67) CDK1PKMCYP2C19GAAALDH1A1
SCHEMBL9714080 0.88 GAA (0.51) CDK1PKMCYP2C19GAAKDM4E
SCHEMBL9713778 0.83 CDK1 (0.68) CDK1PKMCYP2C19GAAKDM4E
SCHEMBL9713935 0.81 PKM (0.67) PKMCYP2C19GAAKDM4EALDH1A1
SCHEMBL9713887 0.81 PKM (0.59) CDK1PKMCYP2C19GAAALDH1A1
SCHEMBL17779214 0.80 PKM (0.70) PKMCYP2C19GAAALDH1A1CA1
SCHEMBL9713798 0.79 CDK1 (0.52) CDK1PKMCYP2C19GAAKDM4E
SCHEMBL9713818 0.79 PKM (0.63) PKMCYP2C19GAAALDH1A1CA1
Mono-N-Acetyl Dapsone SCHEMBL10920445 0.78 PKM (1.00) PKMCYP2C19GAAALDH1A1CA1
SCHEMBL9713865 0.78 PKM (0.62) PKMCYP2C19GAAALDH1A1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed