SCHEMBL9714080

SCHEMBL9714080

COC(=O)c1cc(N)ccc1S(=O)(=O)c1ccc(N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.51
CDK1 P06493 1/20 0.51
ALDH1A1 P00352 4/20 0.51
PKM P14618 3/20 0.51
KDM4E B2RXH2 3/20 0.51
HPGD P15428 2/20 0.51
CA2 P00918 3/20 0.49
CYP2C19 P33261 1/20 0.45
TSHR P16473 2/20 0.44
HTR6 P50406 2/20 0.44
LMNA P02545 1/20 0.44
MPO P05164 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
NPC1 O15118 1/20 0.43
CA1 P00915 1/20 0.43
CA5A P35218 1/20 0.43
CA9 Q16790 1/20 0.43
HSD11B1 P28845 1/20 0.42
F2 P00734 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713813 0.88 CDK1 (0.67) GAACDK1ALDH1A1PKMKDM4E
SCHEMBL9713798 0.84 CDK1 (0.52) GAACDK1ALDH1A1PKMKDM4E
SCHEMBL9713812 0.83 PKM (0.49) GAAALDH1A1PKMKDM4EHPGD
SCHEMBL30827404 0.83 CA2 (0.63) GAACDK1ALDH1A1PKMKDM4E
SCHEMBL11226378 0.83 CA2 (0.63) GAACDK1ALDH1A1PKMKDM4E
SCHEMBL7781881 0.83 GAA (0.56) GAACDK1ALDH1A1PKMKDM4E
SCHEMBL9714078 0.82 CA4 (0.46) GAAALDH1A1PKMKDM4EHPGD
SCHEMBL7411337 0.81 GAA (0.54) GAACDK1ALDH1A1PKMKDM4E
SCHEMBL9713938 0.81 HTR6 (0.50) ALDH1A1PKMKDM4ECA2CYP2C19
Hydrochloric Acid SCHEMBL9713979 0.78 HTR6 (0.47) GAAALDH1A1PKMCA2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed
EP-0165422-B1 SUBSTITUTED BIS-(4-AMINOPHENYL)-SULPHONES, THEIR PREPARATION AND THEIR USE AS MEDICINES Dr. Karl Thomae GmbH (DE) 1988-03-09 EP disclosed