SCHEMBL9713818

SCHEMBL9713818

CC(=O)Nc1ccc(S(=O)(=O)c2ccc(N)cc2N(C)C)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.63
CYP2C19 P33261 1/20 0.63
GAA P10253 2/20 0.52
CA1 P00915 3/20 0.49
CA2 P00918 3/20 0.49
CA12 O43570 2/20 0.49
CA9 Q16790 2/20 0.49
NPC1 O15118 1/20 0.47
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
MMP1 P03956 1/20 0.44
MMP2 P08253 1/20 0.44
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
MMP13 P45452 1/20 0.44
TSHR P16473 1/20 0.44
PAX8 Q06710 1/20 0.44
F2 P00734 2/20 0.44
PRSS1 P07477 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713804 0.86 GAA (0.53) PKMCYP2C19GAACA1CA2
SCHEMBL9713990 0.83 HTR6 (0.50) PKMCYP2C19GAACA1CA2
SCHEMBL9713935 0.82 PKM (0.67) PKMCYP2C19GAACA1CA2
SCHEMBL9713853 0.82 PKM (0.67) PKMCYP2C19GAACA1CA2
SCHEMBL9713937 0.81 KMT2A (0.66) PKMGAAKMT2AMEN1LMNA
SCHEMBL17779214 0.81 PKM (0.70) PKMCYP2C19GAACA1CA2
Mono-N-Acetyl Dapsone SCHEMBL10920445 0.79 PKM (1.00) PKMCYP2C19GAACA1CA2
SCHEMBL9713813 0.79 CDK1 (0.67) PKMCYP2C19GAACA1CA2
SCHEMBL9713865 0.79 PKM (0.62) PKMCYP2C19GAACA1CA2
SCHEMBL9713887 0.77 PKM (0.59) PKMCYP2C19GAACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed