SCHEMBL9713804

SCHEMBL9713804

CC(=O)Nc1ccc(S(=O)(=O)c2ccc(N(C)C)cc2N(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.53
PKM P14618 2/20 0.51
CYP2C19 P33261 1/20 0.50
ALDH1A1 P00352 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TSHR P16473 1/20 0.48
IDO1 P14902 1/20 0.47
KMT2A Q03164 3/20 0.47
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA12 O43570 2/20 0.47
CA9 Q16790 2/20 0.47
LMNA P02545 2/20 0.46
MEN1 O00255 2/20 0.46
MMP1 P03956 1/20 0.46
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
MMP13 P45452 1/20 0.46
PAX8 Q06710 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713818 0.86 PKM (0.63) GAAPKMCYP2C19ALDH1A1L3MBTL1
SCHEMBL9713937 0.83 KMT2A (0.66) GAAPKMALDH1A1KMT2ALMNA
SCHEMBL9713845 0.77 HTR6 (0.46) PKMCYP2C19ALDH1A1TSHRKMT2A
Acedapsone SCHEMBL152710 0.74 PKM (0.85) GAAPKMCYP2C19ALDH1A1L3MBTL1
SCHEMBL59093 0.74 SMN1; SMN2 (0.61) GAACYP2C19ALDH1A1L3MBTL1TSHR
SCHEMBL9714044 0.73 ALDH1A1 (0.59) GAAPKMALDH1A1L3MBTL1TSHR
Acedapsone SCHEMBL28716352 0.73 PKM (0.82) GAAPKMCYP2C19ALDH1A1L3MBTL1
Acedapsone SCHEMBL22518385 0.73 PKM (0.82) GAAPKMCYP2C19ALDH1A1L3MBTL1
Acedapsone SCHEMBL28254874 0.70 PKM (0.72) GAAPKMCYP2C19ALDH1A1L3MBTL1
SCHEMBL9713935 0.69 PKM (0.67) GAAPKMCYP2C19ALDH1A1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed