SCHEMBL9714322

SCHEMBL9714322

CC(c1c(F)cccc1F)n1cnc(C(N)=O)c1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADA P00813 11/20 0.48
CA5A P35218 1/20 0.40
SCN9A Q15858 2/20 0.34
KDM5A P29375 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10568392 0.81 CYP1A2 (0.44)
SCHEMBL24268206 0.75 ADA (0.53) ADAKDM5A
SCHEMBL10959131 0.75 CA5A (0.52) CA5ACES2CES1
SCHEMBL30582304 0.72 CA5A (0.48) ADACA5ASCN9ACES2CES1
SCHEMBL27781574 0.70 ADA (0.51) ADAKDM5A
SCHEMBL9714477 0.69 ALDH1A1 (0.49) CES2CES1
SCHEMBL9714146 0.69 CA5A (0.58) ADACA5AKDM5AKDM5B
SCHEMBL4981212 0.68 ADA (0.55) ADA
SCHEMBL30582364 0.68 ADA (0.43) ADACA5A
SCHEMBL7452973 0.67 ADA (0.48) ADA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0248414-B1 ARALKYL IMIDAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1992-09-23 EP claimed
EP-0248414-A2 Aralkyl imidazole derivatives CIBA-GEIGY AG (CH) 1987-12-09 EP claimed
EP-0248414-B1 ARALKYL IMIDAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1992-09-23 EP disclosed
US-4851424-A 1-Phenyl-lower alkyl-imidazole 4- or 5-carboxamide compounds which are useful in the treatment of epilepsy CIBA-GEIGY CORPORATION (US) 1989-07-25 US disclosed
EP-0248414-A2 Aralkyl imidazole derivatives CIBA-GEIGY AG (CH) 1987-12-09 EP disclosed