SCHEMBL9714477

SCHEMBL9714477

CC(c1c(F)cccc1F)n1cncc1C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
GPBAR1 Q8TDU6 4/20 0.46
MAPK1 P28482 1/20 0.44
GABRA1 P14867 7/20 0.42
GABRB2 P47870 6/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
LMNA P02545 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ABCB11 O95342 1/20 0.42
GABRA2 P47869 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.38
TGFBR1 P36897 3/20 0.34
TGFBR2 P37173 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10569735 0.81 GABRA1 (0.68) ALDH1A1TDP1GPBAR1MAPK1GABRA1
SCHEMBL11733511 0.78 ALDH1A1 (0.78) ALDH1A1TDP1GPBAR1MAPK1GABRA1
SCHEMBL25135971 0.75 ALDH1A1 (0.46) ALDH1A1TDP1GPBAR1MAPK1GABRA1
SCHEMBL9714322 0.69 ADA (0.48) CES2CES1
SCHEMBL11483915 0.69 ALDH1A1 (0.55) ALDH1A1TDP1GPBAR1MAPK1GABRA1
SCHEMBL9714161 0.69 CA5A (0.48) ALDH1A1GPBAR1CYP11B1CYP11B2TGFBR1
SCHEMBL10959131 0.67 CA5A (0.52) ALDH1A1LMNASMN1; SMN2CES2CES1
SCHEMBL1081228 0.66 ALDH1A1 (1.00) ALDH1A1TDP1GPBAR1MAPK1GABRA1
SCHEMBL11726722 0.66 ALDH1A1 (1.00) ALDH1A1TDP1GPBAR1MAPK1GABRA1
SCHEMBL1081229 0.66 ALDH1A1 (1.00) ALDH1A1TDP1GPBAR1MAPK1GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0248414-B1 ARALKYL IMIDAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1992-09-23 EP claimed
EP-0248414-A2 Aralkyl imidazole derivatives CIBA-GEIGY AG (CH) 1987-12-09 EP claimed
EP-0248414-B1 ARALKYL IMIDAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1992-09-23 EP disclosed
US-4851424-A 1-Phenyl-lower alkyl-imidazole 4- or 5-carboxamide compounds which are useful in the treatment of epilepsy CIBA-GEIGY CORPORATION (US) 1989-07-25 US disclosed
EP-0248414-A2 Aralkyl imidazole derivatives CIBA-GEIGY AG (CH) 1987-12-09 EP disclosed