SCHEMBL971460

SCHEMBL971460

COCC(=O)Nc1ccc(Br)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 7/20 1.00
ALDH1A1 P00352 5/20 0.69
MEN1 O00255 4/20 0.66
KMT2A Q03164 4/20 0.66
SMN1; SMN2 Q16637 4/20 0.65
MAPT P10636 3/20 0.65
ALOX12 P18054 1/20 0.65
MAPK1 P28482 1/20 0.65
HTT P42858 1/20 0.65
RAB9A P51151 3/20 0.59
TDP1 Q9NUW8 1/20 0.57
CYP2C19 P33261 1/20 0.56
NPC1 O15118 2/20 0.55
THRB P10828 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14962804 0.90 HPGD (0.81) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL1976948 0.83 HPGD (0.71) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL764569 0.83 HPGD (0.71) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL22854085 0.83 HPGD (0.71) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL6607271 0.82 ALDH1A1 (0.71) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL29349031 0.82 HPGD (0.71) HPGDMEN1KMT2ASMN1; SMN2MAPT
SCHEMBL5206026 0.81 HPGD (0.75) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL2098410 0.81 MTNR1A (0.70) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL2091479 0.81 HPGD (0.70) HPGDALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL853933 0.81 HPGD (0.70) HPGDALDH1A1KMT2ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4539840-A1 KINASE MODULATORS AND METHODS OF USE THEREOF Neuron23, Inc. (US) 2025-04-23 EP disclosed
CN-119730846-A Kinase modulators and methods of use thereof 神经元23公司 2025-03-28 CN disclosed
WO-2023244788-A9 KINASE MODULATORS AND METHODS OF USE THEREOF NEURON23, INC. (US) 2024-09-12 WO disclosed
US-20240025906-A1 KINASE MODULATORS AND METHODS OF USE THEREOF SUNDANCE BIOSCIENCES, INC. 2024-01-25 US disclosed
US-20240025906-A1 KINASE MODULATORS AND METHODS OF USE THEREOF SUNDANCE BIOSCIENCES, INC. 2024-01-25 US disclosed
WO-2023244788-A1 KINASE MODULATORS AND METHODS OF USE THEREOF NEURON23, INC. (US) 2023-12-21 WO disclosed
EP-3421467-A1 5-PHENYLAZAINDOLE DERIVATIVE HAVING AMPK ACTIVATING EFFECT Shionogi & Co., Ltd (JP) 2019-01-02 EP disclosed
WO-2017146186-A1 5-PHENYLAZAINDOLE DERIVATIVE HAVING AMPK ACTIVATING EFFECT 塩野義製薬株式会社 2017-08-31 WO disclosed
US-7871982-B2 Lincomycin derivatives and antimicrobial agents comprising the same as active ingredient MEIJI SEIKA KAISHA, LTD. (JP) 2011-01-18 US disclosed
US-20090156512-A1 potent activity against resistant pneumococci MEIJI SEIKA KAISHA, LTD. (JP) 2009-06-18 US disclosed
EP-1970377-A1 LINCOMYCIN DERIVATIVE AND ANTIBACTERIAL AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT MEIJI SEIKA KAISHA LTD. (JP) 2008-09-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156512-A1 potent activity against resistant pneumococci H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, NAT1, NPM1 HPGD 2051/4885ALDH1A1 2976/4885MEN1 299/4885
US-20240025906-A1 KINASE MODULATORS AND METHODS OF USE THEREOF TYK2, JAK1, JAK3 HPGD 3842/4885ALDH1A1 4807/4885MEN1 3601/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.