SCHEMBL9714665

SCHEMBL9714665

CC(C#N)COc1cccc(CCl)c1.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SGMS2 Q8NHU3 1/20 0.39
MAOB P27338 5/20 0.38
BCHE P06276 4/20 0.38
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TSHR P16473 2/20 0.37
SLC22A2 O15244 1/20 0.37
SLC22A1 O15245 1/20 0.37
SLC22A3 O75751 1/20 0.37
ESR1 P03372 1/20 0.37
CHRM2 P08172 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
CHRM1 P11229 1/20 0.37
DRD2 P14416 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
CHRM3 P20309 1/20 0.37
DRD1 P21728 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714712 0.89 TSHR (0.36) SGMS2MAOBBCHEALDH1A1SMN1; SMN2
SCHEMBL9714816 0.82 SLC6A2 (0.34) MAOBTSHRSLC6A2SLC6A3MEN1
SCHEMBL29463763 0.81 BCHE (0.54) MAOBBCHEALDH1A1MEN1KMT2A
SCHEMBL28703047 0.81 BCHE (0.54) MAOBBCHEALDH1A1MEN1KMT2A
SCHEMBL9714805 0.81 GUSB (0.38) SGMS2
SCHEMBL9714646 0.80 MEN1 (0.35) TSHROPRM1OPRD1MEN1KMT2A
SCHEMBL5973608 0.77 SIGMAR1 (0.53) MAOBALDH1A1SMN1; SMN2CHRM2HTR1A
SCHEMBL9714823 0.77 MAOA (0.35) MAOB
SCHEMBL9714779 0.76 CYP3A4 (0.33) SGMS2MAOBALDH1A1TSHRSLC6A2
Hydrochloric Acid SCHEMBL9714667 0.76 SGMS2 (0.40) SGMS2MAOBBCHEMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166210-A QUINOLINE DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1992-11-24 US disclosed
US-5028615-A Treatment of hypersensitivity RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-07-02 US disclosed
US-4920133-A Quinoline derivatives and use thereof as antagonists of leukotriene D4 RORER PHARMACEUTICAL CORP. (US) 1990-04-24 US disclosed