SCHEMBL9714712

SCHEMBL9714712

CC(C#N)CCOc1cccc(CCl)c1.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.36
MAPK1 P28482 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
SIGMAR1 Q99720 1/20 0.35
SGMS2 Q8NHU3 1/20 0.35
SLC2A1 P11166 1/20 0.34
CTSB P07858 1/20 0.34
BCHE P06276 1/20 0.33
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NR1H4 Q96RI1 1/20 0.33
SLC22A2 O15244 1/20 0.33
SLC22A1 O15245 1/20 0.33
SLC22A3 O75751 1/20 0.33
ESR1 P03372 1/20 0.33
CHRM2 P08172 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
ADORA3 P0DMS8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714665 0.89 SGMS2 (0.39) TSHRTDP1SGMS2BCHEALDH1A1
SCHEMBL9714791 0.87 LTA4H (0.36) MAPK1L3MBTL1TDP1SIGMAR1SLC2A1
SCHEMBL9714805 0.83 GUSB (0.38) SGMS2
SCHEMBL9714646 0.82 MEN1 (0.35) TSHRTDP1OPRM1OPRD1KDM4E
SCHEMBL9714816 0.79 SLC6A2 (0.34) TSHRTDP1SIGMAR1CTSBSLC6A2
Hydrochloric Acid SCHEMBL9714716 0.76 SIGMAR1 (0.39) TSHRMAPK1L3MBTL1TDP1SIGMAR1
SCHEMBL28703047 0.76 BCHE (0.54) L3MBTL1BCHEALDH1A1MAOBKDM4E
SCHEMBL29463763 0.76 BCHE (0.54) L3MBTL1BCHEALDH1A1MAOBKDM4E
SCHEMBL9714829 0.75 CYP3A4 (0.34) TSHRTDP1ALDH1A1KDM4EMEN1
SCHEMBL5973608 0.74 SIGMAR1 (0.53) SIGMAR1ALDH1A1SMN1; SMN2CHRM2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166210-A QUINOLINE DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1992-11-24 US disclosed
US-5028615-A Treatment of hypersensitivity RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-07-02 US disclosed