SCHEMBL9714950

SCHEMBL9714950

Nc1n[nH]c(-c2ccccc2)c1CC(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
RPS6KA3 P51812 1/20 0.49
GAA P10253 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 2/20 0.45
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ILK Q13418 1/20 0.43
PIK3CD O00329 3/20 0.42
PIK3CA P42336 3/20 0.42
PIK3CB P42338 3/20 0.42
PIK3CG P48736 3/20 0.42
PRKDC P78527 3/20 0.42
CYP1A2 P05177 1/20 0.41
LMNA P02545 2/20 0.41
ABCC4 O15439 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714985 0.86 ABL1 (0.43) MAPK1NPSR1RPS6KA3GAASMN1; SMN2
SCHEMBL11242632 0.82 KDM4E (0.50) NPSR1GAASMN1; SMN2KDM4ENPC1
SCHEMBL9714918 0.82 LMNA (0.54) MAPK1NPSR1GAASMN1; SMN2KDM4E
Hydrochloric Acid SCHEMBL9715094 0.81 LMNA (0.53) MAPK1NPSR1GAASMN1; SMN2KDM4E
SCHEMBL9714922 0.80 ALDH1A1 (0.44) MAPK1NPSR1RPS6KA3SMN1; SMN2KDM4E
SCHEMBL9714945 0.78 HSD17B10 (0.46) MAPK1NPSR1GAASMN1; SMN2KDM4E
SCHEMBL2949076 0.71 KDM4E (0.68) MAPK1NPSR1RPS6KA3GAASMN1; SMN2
SCHEMBL5820038 0.70 MAPK1 (1.00) MAPK1NPSR1RPS6KA3GAASMN1; SMN2
SCHEMBL2870468 0.68 GAA (0.68) MAPK1NPSR1RPS6KA3GAASMN1; SMN2
SCHEMBL2875437 0.68 MAPK1 (0.63) MAPK1NPSR1RPS6KA3GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992018484-A1 3-AMINO-5-ARYLPYRAZOLE-4-ACETIC ACID DERIVATIVES EXHIBITING THERAPEUTIC EFFECTS A.H. ROBINS COMPANY, INCORPORATED (US) 1992-10-29 WO claimed
US-5057534-A Anxiolytic, anticonfulsant and muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1991-10-15 US claimed
WO-1992018484-A1 3-AMINO-5-ARYLPYRAZOLE-4-ACETIC ACID DERIVATIVES EXHIBITING THERAPEUTIC EFFECTS A.H. ROBINS COMPANY, INCORPORATED (US) 1992-10-29 WO disclosed
US-5057534-A Anxiolytic, anticonfulsant and muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1991-10-15 US disclosed