SCHEMBL9719015

SCHEMBL9719015

CCCOc1c(Br)cc(C(C#N)(CCC(C#N)(C(=O)OCC)c2cc(OC)c(OC)c(OC)c2)C(=O)OCC)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
HPGD P15428 2/20 0.42
HTT P42858 1/20 0.42
KDM4E B2RXH2 3/20 0.36
PKM P14618 1/20 0.36
TNFRSF1A P19438 1/20 0.35
CNR2 P34972 2/20 0.35
PTAFR P25105 1/20 0.35
POLB P06746 1/20 0.35
NCOA1 Q15788 1/20 0.34
NCOA3 Q9Y6Q9 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9719059 0.86 ALDH1A1 (0.34) ALDH1A1SMN1; SMN2MAPTRAB9AL3MBTL1
SCHEMBL9719050 0.82 KMT2A (0.41) ALDH1A1MAPTL3MBTL1MEN1KMT2A
SCHEMBL9719055 0.81 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2MAPTRAB9AL3MBTL1
SCHEMBL9719109 0.74 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2MAPTRAB9AL3MBTL1
SCHEMBL9719027 0.71 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2MAPTRAB9AL3MBTL1
SCHEMBL3007307 0.69 L3MBTL1 (0.46) ALDH1A1SMN1; SMN2MAPTL3MBTL1MEN1
SCHEMBL28484877 0.66 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL9719008 0.65 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2MAPTRAB9AL3MBTL1
SCHEMBL16751953 0.64 CCR1 (0.37) MAPTRAB9AMEN1KMT2AKDM4E
SCHEMBL12428001 0.63 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2MAPTRAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132463-A Cardiovascular, skin, kidney, respiratory system, and gastrointestinal disorders MERCK & CO., INC. (US) 1992-07-21 US disclosed
EP-0257921-B1 NEW 1,3-DIARYL CYCLOPENTANES AND DERIVATIVES THEREOF AS PAF ANTAGONISTS MERCK & CO. INC. (US) 1992-04-15 EP disclosed
US-5047420-A Platelet activating factor MERCK & CO., INC. (US) 1991-09-10 US disclosed
EP-0257921-A2 New 1,3-diaryl cyclopentanes and derivatives thereof as paf antagonists MERCK & CO. INC. (US) 1988-03-02 EP disclosed