SCHEMBL9719008

SCHEMBL9719008

CCCOc1c(Br)cc(CC#N)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
MEN1 O00255 2/20 0.51
HPGD P15428 2/20 0.51
KMT2A Q03164 2/20 0.51
HTT P42858 2/20 0.51
MAPT P10636 1/20 0.49
RAB9A P51151 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
LMNA P02545 1/20 0.46
HSD17B10 Q99714 2/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
S1PR2 O95136 6/20 0.43
S1PR1 P21453 6/20 0.43
S1PR3 Q99500 5/20 0.43
LPAR2 Q9HBW0 5/20 0.43
S1PR4 O95977 2/20 0.43
S1PR5 Q9H228 1/20 0.43
MITF O75030 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27936092 0.85 CA1 (0.47) ALDH1A1SMN1; SMN2HPGDHTTMAPT
SCHEMBL9718999 0.81 HSD17B10 (0.65) ALDH1A1SMN1; SMN2MEN1HPGDKMT2A
SCHEMBL9719016 0.81 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2MEN1HPGDKMT2A
SCHEMBL1020821 0.76 PTGS2 (0.57) MAPT
SCHEMBL15506125 0.74 PIK3CD (0.37) ALDH1A1HTTMAPTRAB9ALMNA
SCHEMBL6897446 0.74 ALOX5 (0.53) ALDH1A1MEN1KMT2AHTTMAPT
SCHEMBL7281740 0.72 DHFR (0.49) ALDH1A1SMN1; SMN2MEN1KMT2AKDM4E
SCHEMBL4291750 0.71 HSD17B10 (0.60) ALDH1A1SMN1; SMN2MEN1HPGDKMT2A
SCHEMBL4295742 0.71 S1PR2 (0.57) ALDH1A1SMN1; SMN2MEN1HPGDKMT2A
SCHEMBL19818498 0.71 PTGS2 (0.67) ALDH1A1SMN1; SMN2MEN1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132463-A Cardiovascular, skin, kidney, respiratory system, and gastrointestinal disorders MERCK & CO., INC. (US) 1992-07-21 US disclosed
EP-0257921-B1 NEW 1,3-DIARYL CYCLOPENTANES AND DERIVATIVES THEREOF AS PAF ANTAGONISTS MERCK & CO. INC. (US) 1992-04-15 EP disclosed
US-5047420-A Platelet activating factor MERCK & CO., INC. (US) 1991-09-10 US disclosed
EP-0257921-A2 New 1,3-diaryl cyclopentanes and derivatives thereof as paf antagonists MERCK & CO. INC. (US) 1988-03-02 EP disclosed