SCHEMBL9720563

SCHEMBL9720563

CCC(=O)c1ccc(Cl)c(C)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 1/20 0.44
CYP3A4 P08684 1/20 0.41
POLB P06746 3/20 0.38
SHBG P04278 1/20 0.37
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CRHR1 P34998 1/20 0.36
MAPK1 P28482 1/20 0.36
HIF1A Q16665 1/20 0.36
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
TSHR P16473 1/20 0.35
LMNA P02545 1/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8105720 0.83 HSP90AB1 (0.41) HSP90AB1CYP3A4POLBSHBGRAB9A
SCHEMBL18535886 0.83 HSP90AB1 (0.41) HSP90AB1CYP3A4POLBSHBGRAB9A
SCHEMBL28159519 0.82 LMNA (0.46) CYP3A4POLBRAB9AALDH1A1KDM4E
SCHEMBL7450427 0.79 HSP90AB1 (0.47) HSP90AB1POLBALDH1A1KDM4EMEN1
SCHEMBL11574084 0.78 HSP90AB1 (0.43) HSP90AB1POLBALDH1A1KDM4EMEN1
SCHEMBL15133627 0.78 NPC1 (0.40) HSP90AB1POLBRAB9AKDM4EMEN1
SCHEMBL28385050 0.78 HSP90AB1 (0.46) HSP90AB1CYP3A4POLBALDH1A1KDM4E
SCHEMBL30093973 0.77 CYP4F2 (0.55) ALDH1A1MEN1KMT2AMAPK1CYP4F2
SCHEMBL9712335 0.77 ALDH1A1 (0.38) CYP3A4ALDH1A1KDM4EMEN1KMT2A
SCHEMBL27544752 0.77 CSNK2A2 (0.49) CYP3A4POLBRAB9AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5103022-A Reacting dl-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino -1-propanone with l-acetylphenylglycine to form corresponding diastereomeric salt, deposition, isolation of l-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino-1-propanone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1992-04-07 US disclosed
US-5057535-A Muscle relaxants NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1991-10-15 US disclosed
EP-0200942-A2 New derivatives of an aminoketone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1986-11-12 EP disclosed