SCHEMBL9720580

SCHEMBL9720580

CCC(=O)c1ccc(OC)c2c1CCC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.47
ADRA1A P35348 1/20 0.41
MTNR1A P48039 3/20 0.40
MTNR1B P49286 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HPGDS O60760 1/20 0.40
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
STAT6 P42226 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9576976 0.97 HMGCR (0.47) HMGCRADRA1AMTNR1AMTNR1BALDH1A1
SCHEMBL12567492 0.85 ADRA1A (0.41) ADRA1AMTNR1AMTNR1BALDH1A1MEN1
SCHEMBL9576702 0.84 ALDH1A1 (0.47) HMGCRADRA1AMTNR1AMTNR1BALDH1A1
SCHEMBL12565602 0.83 ALDH1A1 (0.50) ADRA1AMTNR1AMTNR1BALDH1A1TDP1
SCHEMBL17874456 0.83 DPP4 (0.47) MTNR1AMTNR1BALDH1A1MEN1KMT2A
SCHEMBL12918718 0.80 HTT (0.52) ALDH1A1MEN1KMT2APOLBRXRA
SCHEMBL3427457 0.79 ALDH1A1 (0.50) ADRA1AALDH1A1TDP1L3MBTL1CYP3A4
SCHEMBL3424668 0.79 MAPT (0.50) ADRA1AALDH1A1TDP1RXRARXRB
SCHEMBL833885 0.78 ADRA1A (0.59) ADRA1AALDH1A1CA9KDM4EGLA
SCHEMBL9720538 0.77 ALDH1A1 (0.41) ADRA1AALDH1A1MEN1KMT2ARXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5103022-A Reacting dl-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino -1-propanone with l-acetylphenylglycine to form corresponding diastereomeric salt, deposition, isolation of l-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino-1-propanone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1992-04-07 US disclosed
US-5057535-A Muscle relaxants NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1991-10-15 US disclosed
EP-0200942-A2 New derivatives of an aminoketone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1986-11-12 EP disclosed