SCHEMBL9720538

SCHEMBL9720538

COc1ccc(C(=O)CCCCl)c2c1CCCC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
STAT6 P42226 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
RXRA P19793 4/20 0.38
RXRB P28702 4/20 0.38
RXRG P48443 4/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC8 Q9BY41 1/20 0.38
THRA P10827 2/20 0.38
THRB P10828 2/20 0.38
ADRA1A P35348 1/20 0.37
RBP1 P09455 1/20 0.37
HTR4 Q13639 1/20 0.37
MIF P14174 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9576702 0.84 ALDH1A1 (0.47) ALDH1A1CYP1A2CYP3A4CYP2C9STAT6
SCHEMBL12918718 0.82 HTT (0.52) ALDH1A1CYP1A2CYP3A4CYP2C9STAT6
SCHEMBL12567492 0.82 ADRA1A (0.41) ALDH1A1CYP1A2CYP3A4CYP2C9STAT6
SCHEMBL9720624 0.81 LMNA (0.56) ALDH1A1MEN1KMT2AHTR4HTR2A
SCHEMBL9576976 0.80 HMGCR (0.47) ALDH1A1CYP1A2CYP3A4CYP2C9STAT6
SCHEMBL10657187 0.78 THRB (0.50) ALDH1A1CYP1A2CYP3A4CYP2C9STAT6
SCHEMBL4255074 0.78 PDE4D (0.53) ALDH1A1MEN1KMT2A
SCHEMBL9720580 0.77 HMGCR (0.47) ALDH1A1CYP1A2CYP3A4CYP2C9STAT6
SCHEMBL3427457 0.77 ALDH1A1 (0.50) ALDH1A1CYP3A4HSD17B10ADRA1ARBP1
SCHEMBL3424668 0.77 MAPT (0.50) ALDH1A1RXRARXRBRXRGADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5103022-A Reacting dl-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino -1-propanone with l-acetylphenylglycine to form corresponding diastereomeric salt, deposition, isolation of l-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino-1-propanone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1992-04-07 US disclosed
US-5057535-A Muscle relaxants NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1991-10-15 US disclosed
EP-0200942-A2 New derivatives of an aminoketone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1986-11-12 EP disclosed