SCHEMBL9724124

SCHEMBL9724124

Cc1nc2ccc(CBr)cc2c(Cl)c1Br

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2D6 P10635 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
KDM4E B2RXH2 1/20 0.43
CYP3A4 P08684 1/20 0.43
HIF1A Q16665 1/20 0.43
PKM P14618 1/20 0.41
ALDH1A1 P00352 5/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 2/20 0.37
MEN1 O00255 1/20 0.37
RAD52 P43351 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724276 0.87 CYP2C19 (0.48) CYP2C19CYP1A2CYP2C9CYP2D6RXFP1
SCHEMBL9724301 0.86 CYP2C19 (0.50) CYP2C19CYP1A2CYP2C9CYP2D6RXFP1
SCHEMBL9724155 0.80 LMNA (0.51) CYP2C19CYP1A2CYP2C9CYP2D6RXFP1
SCHEMBL10517897 0.78 CYP1A2 (0.48) CYP2C19CYP1A2CYP2C9CYP2D6RXFP1
SCHEMBL9380126 0.74 LMNA (0.62) CYP2C19CYP1A2CYP2C9CYP2D6RXFP1
SCHEMBL2539722 0.74 KDM4E (0.76) CYP2C19CYP1A2CYP2C9CYP2D6RXFP1
SCHEMBL4421151 0.73 HTT (0.41) CYP2C19CYP1A2CYP2C9CYP2D6RXFP1
SCHEMBL12877168 0.73 MAOA (0.57) CYP2C19CYP1A2CYP2C9CYP2D6RXFP1
SCHEMBL9724225 0.72 ALDH1A1 (0.39) CYP2C19CYP1A2KDM4ECYP3A4HIF1A
SCHEMBL9724241 0.72 KDM4E (0.50) CYP2C19CYP1A2CYP2C9CYP2D6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed