SCHEMBL9724227

SCHEMBL9724227

Cc1ccc2nc(CF)cc(Cl)c2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.62
KDM4E B2RXH2 3/20 0.43
MAPT P10636 2/20 0.43
ALDH1A1 P00352 2/20 0.43
PKM P14618 1/20 0.40
ELANE P08246 3/20 0.39
ACHE P22303 5/20 0.38
BCHE P06276 4/20 0.38
GRIN1 Q05586 4/20 0.38
GRIN2A Q12879 4/20 0.38
NT5E P21589 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724146 0.85 LMNA (0.64) LMNAKDM4EMAPTALDH1A1PKM
SCHEMBL9494320 0.85 LMNA (0.64) LMNAKDM4EMAPTALDH1A1PKM
SCHEMBL9724121 0.83 LMNA (0.62) LMNAKDM4EMAPTALDH1A1PKM
SCHEMBL16256881 0.81 ALDH1A1 (0.40) LMNAKDM4EMAPTALDH1A1NT5E
SCHEMBL9724211 0.78 NT5E (0.39) LMNAKDM4ENT5E
SCHEMBL4768081 0.77 LMNA (1.00) LMNAKDM4EMAPTALDH1A1PKM
SCHEMBL30572382 0.77 LMNA (1.00) LMNAKDM4EMAPTALDH1A1PKM
SCHEMBL829490 0.77 LMNA (0.72) LMNAKDM4EMAPTALDH1A1PKM
Hydrochloric Acid SCHEMBL9494656 0.75 LMNA (0.96) LMNAKDM4EMAPTALDH1A1ELANE
SCHEMBL9724150 0.75 LMNA (0.51) LMNAKDM4EMAPTALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed