SCHEMBL9725103

SCHEMBL9725103

NCCN1CCN(c2cc(C(F)(F)F)ccn2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.59
KDM4E B2RXH2 3/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
CYP2D6 P10635 1/20 0.53
PPARG P37231 1/20 0.48
PPARD Q03181 1/20 0.48
PPARA Q07869 1/20 0.48
DRD2 P14416 1/20 0.47
DRD1 P21728 1/20 0.47
DRD3 P35462 1/20 0.47
FFAR4 Q5NUL3 1/20 0.46
MAPT P10636 3/20 0.46
ALDH1A1 P00352 3/20 0.45
LMNA P02545 1/20 0.45
HSD17B10 Q99714 1/20 0.45
PARP1 P09874 1/20 0.44
TRPV1 Q8NER1 2/20 0.43
PIK3C3 Q8NEB9 1/20 0.43
TSHR P16473 1/20 0.43
DPP4 P27487 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971652 0.83 ADRB1 (0.62) ADRB1KDM4EL3MBTL1CYP2D6PPARG
SCHEMBL12968838 0.81 ADRB1 (0.68) ADRB1KDM4EL3MBTL1CYP2D6PPARG
SCHEMBL18176129 0.79 ADRB1 (0.73) ADRB1KDM4EL3MBTL1CYP2D6PPARG
SCHEMBL3140922 0.78 DRD4 (0.53) DRD2DRD3ALDH1A1PIK3C3DPP4
SCHEMBL7130750 0.78 ADRB1 (0.59) ADRB1KDM4EL3MBTL1CYP2D6FFAR4
SCHEMBL24008459 0.77 ADRB1 (0.71) ADRB1KDM4EL3MBTL1CYP2D6PPARG
SCHEMBL31061118 0.76 CXCR3 (0.52) ADRB1KDM4EL3MBTL1CYP2D6PPARG
SCHEMBL2799020 0.76 ADRA1B (0.52) ADRB1KDM4EL3MBTL1CYP2D6DRD2
SCHEMBL1901605 0.76 ADRB1 (0.69) ADRB1KDM4EL3MBTL1CYP2D6PPARG
SCHEMBL1998032 0.76 ADRB1 (0.69) ADRB1KDM4EL3MBTL1CYP2D6PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135931-A Antidepressants, psychological disorders, nervous system disorders AKZO N.V. (NL) 1992-08-04 US disclosed
EP-0462638-A1 Pyridinylpiperazine derivatives Akzo Nobel N.V. (NL) 1991-12-27 EP disclosed