SCHEMBL9726474

SCHEMBL9726474

Cn1nnnc1C=C(c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.41
CYP11B2 P19099 2/20 0.41
TDP1 Q9NUW8 2/20 0.40
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HSP90AA1 P07900 1/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HIF1A Q16665 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
PTGS2 P35354 1/20 0.36
CYP2D6 P10635 1/20 0.35
ESR1 P03372 1/20 0.34
ALDH1A1 P00352 2/20 0.34
HSD11B1 P28845 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726766 0.91 PTGS2 (0.44) CYP19A1CYP11B2TDP1MAPTKDM4E
SCHEMBL9726776 0.91 PTGS2 (0.44) CYP19A1CYP11B2TDP1MAPTKDM4E
SCHEMBL9726773 0.91 PTGS2 (0.44) CYP19A1CYP11B2TDP1MAPTKDM4E
SCHEMBL9727011 0.81 ALDH1A1 (0.51) TDP1MAPTKDM4EGAARAB9A
SCHEMBL8999117 0.71 PTGS2 (0.39) CYP19A1CYP11B2TDP1MAPTKDM4E
SCHEMBL9726825 0.70 ALDH1A1 (0.39) TDP1HTTRAB9AALDH1A1MEN1
Hydrochloric Acid SCHEMBL11510394 0.68 MAPT (0.33) TDP1MAPTKDM4EHSP90AA1GAA
SCHEMBL10131999 0.67 MAPT (0.40) TDP1MAPTKDM4EHSP90AA1GAA
SCHEMBL15174968 0.66 TDP1 (0.39) TDP1MAPTKDM4EHSP90AA1GAA
SCHEMBL9726944 0.65 HMGCR (0.42) TDP1MAPTKDM4EHSP90AA1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4898949-A Intermediates for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-02-06 US claimed
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4939265-A Intermediates and process for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-07-03 US disclosed
US-4898949-A Intermediates for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-02-06 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed