SCHEMBL9727011

SCHEMBL9727011

COc1ccc(C(=Cc2nnnn2C)c2ccc(OC)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
KDM4E B2RXH2 2/20 0.51
MAPT P10636 1/20 0.51
HPGD P15428 1/20 0.51
TDP1 Q9NUW8 1/20 0.40
MGAM O43451 1/20 0.39
F12 P00748 1/20 0.39
AMY1A P0DUB6 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
NQO2 P16083 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726773 0.77 PTGS2 (0.44) ALDH1A1KDM4EMAPTHPGDTDP1
SCHEMBL9726766 0.77 PTGS2 (0.44) ALDH1A1KDM4EMAPTHPGDTDP1
SCHEMBL9726776 0.77 PTGS2 (0.44) ALDH1A1KDM4EMAPTHPGDTDP1
SCHEMBL10385010 0.72 NQO2 (0.43) ALDH1A1KDM4EMAPTHPGDTDP1
SCHEMBL10385011 0.72 NQO2 (0.43) ALDH1A1KDM4EMAPTHPGDTDP1
SCHEMBL4683697 0.71 ALDH1A1 (0.49) ALDH1A1KDM4EMAPTHPGDGAA
SCHEMBL10425548 0.71 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTTDP1MGAM
SCHEMBL9839256 0.69 ALDH1A1 (1.00) ALDH1A1KDM4EMAPTHPGDPDE4A
SCHEMBL9726963 0.69 TCF4 (0.46) ALDH1A1KDM4EMAPTHPGDTDP1
SCHEMBL4685242 0.69 ALDH1A1 (0.45) ALDH1A1KDM4ETDP1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4939265-A Intermediates and process for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-07-03 US disclosed
US-4898949-A Intermediates for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-02-06 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed