SCHEMBL9726545

SCHEMBL9726545

CCCOc1cc(CNc2cnn(CC)c(=O)c2Br)ccc1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.41
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KMT2A Q03164 3/20 0.38
THRB P10828 2/20 0.38
MEN1 O00255 2/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 5/20 0.38
MAPT P10636 4/20 0.38
LMNA P02545 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
APAF1 O14727 1/20 0.38
JAK3 P52333 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
PDE4A P27815 2/20 0.37
MAPK1 P28482 2/20 0.37
PDE4D Q08499 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726550 0.89 PDE5A (0.41) PDE5AHTTNPSR1KMT2ATHRB
SCHEMBL9726466 0.88 PDE5A (0.41) PDE5AHTTNPSR1KMT2ATHRB
SCHEMBL9726673 0.88 BRD4 (0.46) PDE5AHTTNPSR1KMT2APOLB
SCHEMBL9726652 0.86 THRB (0.39) HTTNPSR1KMT2ATHRBMEN1
SCHEMBL9726418 0.81 KDM4E (0.46) PDE5AHTTKMT2ATHRBMEN1
SCHEMBL9726489 0.80 ALDH1A1 (0.46) PDE5AHTTKMT2ATHRBMEN1
SCHEMBL9726693 0.80 KDM4E (0.45) PDE5AHTTNPSR1KMT2ATHRB
SCHEMBL9827490 0.80 KMT2A (0.49) NPSR1KMT2AMEN1POLBKDM4E
SCHEMBL9726895 0.80 PDE9A (0.45) KMT2AMEN1KDM4EMAPTLMNA
SCHEMBL9726506 0.79 ALDH1A1 (0.44) PDE5AHTTKMT2ATHRBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US claimed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP claimed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP claimed