SCHEMBL9726744

SCHEMBL9726744

CC(C)(C)n1nnc(C(CO)=C(c2ccc(F)cc2)c2ccc(F)cc2)n1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 3/20 0.33
AOC3 Q16853 2/20 0.33
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ESR1 P03372 1/20 0.32
CYP19A1 P11511 1/20 0.32
PTGS2 P35354 1/20 0.31
ESRRG P62508 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726587 0.80 TRPM8 (0.43) ESR2RAB9ASMN1; SMN2
SCHEMBL9726796 0.77 HMGCR (0.32) AOC3RAB9ASMN1; SMN2PTGS2
SCHEMBL9726463 0.74 HSD17B10 (0.39) RAB9ASMN1; SMN2
SCHEMBL9726583 0.74 SMN1; SMN2 (0.38) RAB9ASMN1; SMN2
SCHEMBL9726494 0.74 HMGCR (0.32) AOC3
SCHEMBL9726501 0.74 HMGCR (0.32) AOC3
SCHEMBL9726990 0.73 CES2 (0.40) AOC3RAB9ASMN1; SMN2PTGS2
SCHEMBL10612239 0.69 CYP1A2 (0.40) RAB9ASMN1; SMN2
SCHEMBL10612229 0.69 AOC3 (0.30) AOC3
SCHEMBL9726535 0.68 HMGCR (0.46) ESR2RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed