SCHEMBL9726990

SCHEMBL9726990

C=C(C(=O)c1ccc(F)cc1)c1nnn(C(C)(C)C)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.34
RAB9A P51151 2/20 0.34
PTGS2 P35354 1/20 0.33
MGAM O43451 1/20 0.33
AMY1A P0DUB6 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
LMNA P02545 2/20 0.32
NPC1 O15118 1/20 0.32
TP53 P04637 1/20 0.32
RECQL P46063 1/20 0.32
HTR2A P28223 1/20 0.31
USP2 O75604 1/20 0.31
HSD17B10 Q99714 1/20 0.31
LTA4H P09960 1/20 0.31
MGLL Q99685 1/20 0.31
CA1 P00915 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10611800 0.82 CES2 (0.36) CES2CES1SMN1; SMN2RAB9AMGAM
SCHEMBL10612239 0.80 CYP1A2 (0.40) SMN1; SMN2RAB9AGAANPC1TP53
SCHEMBL10612229 0.76 AOC3 (0.30) AOC3
SCHEMBL9726796 0.75 HMGCR (0.32) SMN1; SMN2RAB9APTGS2AOC3
SCHEMBL10608803 0.73 LMNA (0.30) LMNA
SCHEMBL9726744 0.73 ESR2 (0.33) SMN1; SMN2RAB9APTGS2AOC3
SCHEMBL9726583 0.72 SMN1; SMN2 (0.38) CES2CES1SMN1; SMN2RAB9AGAA
SCHEMBL9726494 0.71 HMGCR (0.32) AOC3
SCHEMBL9726501 0.71 HMGCR (0.32) AOC3
SCHEMBL9726984 0.69 TRPA1 (0.34) PTGS2LMNAAOC3NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed