SCHEMBL9726796

SCHEMBL9726796

CC(C)(C)n1nnc(C(C=O)=C(c2ccc(F)cc2)c2ccc(F)cc2)n1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.32
AOC3 Q16853 2/20 0.32
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726494 0.88 HMGCR (0.32) HMGCRAOC3
SCHEMBL9726501 0.88 HMGCR (0.32) HMGCRAOC3
SCHEMBL9726434 0.83 HSD11B1 (0.37) HMGCRRAB9ASMN1; SMN2
SCHEMBL9726578 0.83 MGAM (0.32) HMGCR
SCHEMBL9726424 0.82 HMGCR (0.36) HMGCRRAB9ASMN1; SMN2
SCHEMBL9726403 0.79 TRPM8 (0.42) HMGCRRAB9ASMN1; SMN2
SCHEMBL10612222 0.78 AOC3 (0.30) AOC3
SCHEMBL10612229 0.78 AOC3 (0.30) AOC3
SCHEMBL9726744 0.77 ESR2 (0.33) AOC3RAB9ASMN1; SMN2PTGS2
SCHEMBL9726984 0.76 TRPA1 (0.34) AOC3PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed