SCHEMBL9727125

SCHEMBL9727125

COc1ccc(CN2CCC(NC(=O)c3oc4ccccc4c3C)CC2)cc1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.68
MEN1 O00255 1/20 0.68
ALDH1A1 P00352 1/20 0.68
LMNA P02545 1/20 0.68
KMT2A Q03164 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
MCHR1 Q99705 4/20 0.65
DRD4 P21917 2/20 0.64
ACHE P22303 5/20 0.61
SIGMAR1 Q99720 1/20 0.59
NPC1 O15118 3/20 0.59
RAB9A P51151 3/20 0.59
BCHE P06276 3/20 0.57
KCNH2 Q12809 1/20 0.56
MAOB P27338 3/20 0.56
HRH3 Q9Y5N1 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15926024 0.86 MCHR1 (0.67) KDM4EMEN1ALDH1A1LMNAKMT2A
SCHEMBL9727133 0.86 DRD4 (0.66) KDM4EMEN1ALDH1A1LMNAKMT2A
SCHEMBL9727095 0.82 DRD4 (0.72) ALDH1A1SMN1; SMN2MCHR1DRD4ACHE
SCHEMBL9727116 0.82 MAOB (0.73) MCHR1DRD4ACHESIGMAR1KCNH2
SCHEMBL9727091 0.80 DRD4 (0.70) KDM4EALDH1A1MCHR1DRD4ACHE
SCHEMBL9727049 0.79 MAOB (0.80) MCHR1DRD4ACHESIGMAR1KCNH2
SCHEMBL9872559 0.79 DRD4 (0.78) MEN1KMT2ASMN1; SMN2MCHR1DRD4
SCHEMBL1156414 0.79 NPC1 (0.90) MEN1ALDH1A1LMNAKMT2ASMN1; SMN2
SCHEMBL9727136 0.77 DRD4 (0.67) KDM4EALDH1A1DRD4ACHERAB9A
SCHEMBL9852057 0.75 DRD4 (0.67) MEN1ALDH1A1KMT2ASMN1; SMN2MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098915-A Antiarrhythmia agents G. D. SEARLE & CO. (US) 1992-03-24 US claimed