SCHEMBL9727116

SCHEMBL9727116

COc1ccc(CN2CCC(NC(=O)c3coc4ccccc34)CC2)cc1

nearest known ligand 0.73

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOB P27338 9/20 0.73
DRD4 P21917 4/20 0.71
MAOA P21397 1/20 0.61
SIGMAR1 Q99720 2/20 0.60
MCHR1 Q99705 3/20 0.57
ACHE P22303 1/20 0.57
KCNH2 Q12809 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727049 0.93 MAOB (0.80) MAOBDRD4MAOASIGMAR1MCHR1
SCHEMBL9727095 0.83 DRD4 (0.72) MAOBDRD4SIGMAR1MCHR1ACHE
SCHEMBL9727125 0.82 KDM4E (0.68) MAOBDRD4SIGMAR1MCHR1ACHE
SCHEMBL9727136 0.80 DRD4 (0.67) MAOBDRD4ACHE
SCHEMBL9872559 0.80 DRD4 (0.78) DRD4SIGMAR1MCHR1ACHE
SCHEMBL9727091 0.79 DRD4 (0.70) MAOBDRD4SIGMAR1MCHR1ACHE
SCHEMBL9727133 0.79 DRD4 (0.66) MAOBDRD4SIGMAR1MCHR1ACHE
SCHEMBL30569390 0.79 MAOB (0.60) MAOBKCNH2
SCHEMBL9852057 0.76 DRD4 (0.67) DRD4SIGMAR1MCHR1
SCHEMBL9727102 0.76 SIGMAR1 (0.72) DRD4SIGMAR1MCHR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098915-A Antiarrhythmia agents G. D. SEARLE & CO. (US) 1992-03-24 US claimed
EP-0416581-A1 Substituted N-benzylpiperidine amides G.D. Searle & Co. (US) 1991-03-13 EP claimed