SCHEMBL9727133

SCHEMBL9727133

COc1ccc(CN2CCC(NC(=O)c3oc(C)c4ccccc34)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.66
SIGMAR1 Q99720 2/20 0.61
MCHR1 Q99705 5/20 0.58
ACHE P22303 2/20 0.58
KCNH2 Q12809 1/20 0.56
HRH3 Q9Y5N1 1/20 0.56
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
MEN1 O00255 1/20 0.55
LMNA P02545 1/20 0.55
KMT2A Q03164 1/20 0.55
HPGD P15428 1/20 0.55
HSD17B10 Q99714 1/20 0.55
MAOB P27338 2/20 0.54
BCHE P06276 1/20 0.53
CCR3 P51677 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727125 0.86 KDM4E (0.68) DRD4SIGMAR1MCHR1ACHEKCNH2
SCHEMBL9727095 0.84 DRD4 (0.72) DRD4SIGMAR1MCHR1ACHEALDH1A1
SCHEMBL9872559 0.81 DRD4 (0.78) DRD4SIGMAR1MCHR1ACHESMN1; SMN2
SCHEMBL9727116 0.79 MAOB (0.73) DRD4SIGMAR1MCHR1ACHEKCNH2
SCHEMBL9727091 0.78 DRD4 (0.70) DRD4SIGMAR1MCHR1ACHEKCNH2
SCHEMBL9727049 0.77 MAOB (0.80) DRD4SIGMAR1MCHR1ACHEKCNH2
SCHEMBL9852057 0.77 DRD4 (0.67) DRD4SIGMAR1MCHR1ALDH1A1SMN1; SMN2
SCHEMBL9727102 0.77 SIGMAR1 (0.72) DRD4SIGMAR1MCHR1KCNH2HRH3
SCHEMBL5862230 0.76 SIGMAR1 (1.00) SIGMAR1
Iodide SCHEMBL9852255 0.76 DRD4 (0.60) DRD4SIGMAR1MCHR1ACHEKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098915-A Antiarrhythmia agents G. D. SEARLE & CO. (US) 1992-03-24 US claimed