SCHEMBL9727980

SCHEMBL9727980

Nc1nc(-c2cccnc2)c(Cl)s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.51
KDM4E B2RXH2 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
PIK3CD O00329 1/20 0.50
PIP5K1C O60331 1/20 0.50
PIK3CA P42336 1/20 0.50
PI4KA P42356 1/20 0.50
PI4KB Q9UBF8 1/20 0.50
ALDH1A1 P00352 3/20 0.49
MEN1 O00255 2/20 0.49
MAPT P10636 2/20 0.49
KMT2A Q03164 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
CYP2A6 P11509 6/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP2E1 P05181 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2B6 P20813 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2432630 0.80 ALDH1A1 (0.63) KDM4ESMN1; SMN2PIK3CAPI4KAPI4KB
SCHEMBL9727832 0.80 CYP2A6 (0.49) SMN1; SMN2ALDH1A1CYP2A6CYP3A4CYP2D6
SCHEMBL9833618 0.80 SMN1; SMN2 (0.51) TGFBR1KDM4ESMN1; SMN2PIK3CDPIP5K1C
SCHEMBL6545502 0.79 ALDH1A1 (0.72) TGFBR1KDM4ESMN1; SMN2PIK3CDPIP5K1C
SCHEMBL1850222 0.76 ADORA2A (0.54) TGFBR1KDM4ESMN1; SMN2PIK3CDPIP5K1C
SCHEMBL13930450 0.75 PIK3CA (0.52) TGFBR1KDM4ESMN1; SMN2PIK3CDPIK3CA
SCHEMBL9728291 0.73 CYP2A6 (0.42) KDM4ESMN1; SMN2ALDH1A1MEN1MAPT
SCHEMBL27680210 0.72 ADORA3 (0.48) TGFBR1KDM4ESMN1; SMN2PIK3CDPIP5K1C
SCHEMBL19839753 0.72 ALDH1A1 (0.51) TGFBR1KDM4ESMN1; SMN2PIK3CDPIP5K1C
SCHEMBL13910994 0.71 CYP2A6 (0.70) KDM4ESMN1; SMN2ALDH1A1MAPTCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5128340-A Thiazole derivatives AKZO N.V. (NL) 1992-07-07 US disclosed
EP-0372125-A1 Oxazole and thiazole derivatives AKZO N.V. (NL) 1990-06-13 EP disclosed
EP-0368384-A1 Thiazole derivatives AKZO N.V. (NL) 1990-05-16 EP disclosed