SCHEMBL27680210

SCHEMBL27680210

Nc1nc(-c2cccnc2)c(-n2ccnc2)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.48
ADORA2A P29274 3/20 0.48
ADORA1 P30542 3/20 0.48
CYP3A4 P08684 7/20 0.48
CYP1A2 P05177 4/20 0.48
TDP1 Q9NUW8 4/20 0.48
LMNA P02545 4/20 0.48
CYP2D6 P10635 3/20 0.48
TSHR P16473 3/20 0.48
ALDH1A1 P00352 2/20 0.48
HSD17B10 Q99714 2/20 0.48
MAPK1 P28482 1/20 0.48
CYP2A6 P11509 2/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
MAPT P10636 2/20 0.45
TGFBR1 P36897 1/20 0.44
CLK4 Q9HAZ1 2/20 0.44
USP2 O75604 2/20 0.44
HIF1A Q16665 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27699163 0.87 MEN1 (0.51) ADORA3ADORA2AADORA1CYP3A4CYP1A2
SCHEMBL9727980 0.72 TGFBR1 (0.51) ADORA2AADORA1CYP3A4CYP1A2TDP1
SCHEMBL9833618 0.72 SMN1; SMN2 (0.51) CYP3A4CYP1A2TDP1LMNACYP2D6
SCHEMBL7466847 0.71 ADORA1 (0.50) ADORA2AADORA1CYP3A4CYP1A2TDP1
SCHEMBL6545502 0.71 ALDH1A1 (0.72) ADORA2AADORA1CYP3A4CYP1A2TDP1
SCHEMBL27680206 0.70 ALDH1A1 (0.56) ADORA2AADORA1CYP3A4CYP1A2TDP1
SCHEMBL1850222 0.69 ADORA2A (0.54) ADORA2AADORA1CYP3A4TDP1CYP2D6
SCHEMBL7471062 0.67 ABL1 (0.51) ADORA2AADORA1CYP3A4CYP1A2TDP1
SCHEMBL28395564 0.67 LMNA (0.38) ADORA2AADORA1CYP3A4CYP1A2TDP1
SCHEMBL23331514 0.65 CYP3A4 (0.67) CYP3A4CYP1A2TDP1LMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101041657-A Imines derivative of 4,5-disubstituted-2-aminothiazole having anticancer action and preparation thereof UNIV NANKAI (CN) 2007-09-26 CN disclosed